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Breast drug failure cause found | Breast drug failure cause found |
(1 day later) | |
Scientists have identified a key reason for the drug tamoxifen failing to help some women with breast cancer. | Scientists have identified a key reason for the drug tamoxifen failing to help some women with breast cancer. |
The Cancer Research UK team pinpointed a molecular imbalance which stops the drug working. | The Cancer Research UK team pinpointed a molecular imbalance which stops the drug working. |
Writing in Nature, the team say having this detailed understanding will help develop more effective treatments for women with breast cancer. | Writing in Nature, the team say having this detailed understanding will help develop more effective treatments for women with breast cancer. |
The Cambridge researchers add that the finding could also help explain other examples of drug resistance. | The Cambridge researchers add that the finding could also help explain other examples of drug resistance. |
Previously our understanding of why this occurred could be compared with trying to fix a broken car without knowing how the engine worked Dr Jason Carroll, Cambridge Research Institute | Previously our understanding of why this occurred could be compared with trying to fix a broken car without knowing how the engine worked Dr Jason Carroll, Cambridge Research Institute |
Oestrogen can cause breast cancer cells to grow and divide but tamoxifen prevents this, helping lower the risk of the disease returning. | Oestrogen can cause breast cancer cells to grow and divide but tamoxifen prevents this, helping lower the risk of the disease returning. |
Around 45,000 cases of breast cancer are diagnosed in the UK each year - and up to two-thirds will be prescribed the drug. Women ideally take it for five years after their diagnosis. | Around 45,000 cases of breast cancer are diagnosed in the UK each year - and up to two-thirds will be prescribed the drug. Women ideally take it for five years after their diagnosis. |
But 25-30% will develop resistance to the treatment after time, meaning their cancer is more likely to return. | But 25-30% will develop resistance to the treatment after time, meaning their cancer is more likely to return. |
Scientists have been seeking ways of identifying these women so that time is not wasted, and treatment is better tailored. | Scientists have been seeking ways of identifying these women so that time is not wasted, and treatment is better tailored. |
'We can make repairs' | 'We can make repairs' |
In this study, which involved 100 breast cancer patients, the Cancer Research UK Cambridge Research Institute found tamoxifen works by switching off the breast cancer gene HER2 via a protein called PAX2. | In this study, which involved 100 breast cancer patients, the Cancer Research UK Cambridge Research Institute found tamoxifen works by switching off the breast cancer gene HER2 via a protein called PAX2. |
In patients receiving tamoxifen treatment, the highest levels of PAX2 were associated with improved survival. | In patients receiving tamoxifen treatment, the highest levels of PAX2 were associated with improved survival. |
In contrast, tumours resistant to the drug had higher levels of another molecule, AIB-1, which competes with PAX2 in a molecular "tug-of-war" to control HER2. | In contrast, tumours resistant to the drug had higher levels of another molecule, AIB-1, which competes with PAX2 in a molecular "tug-of-war" to control HER2. |
Tamoxifen has been a huge success story helping to prevent breast cancer recurring for many women Professor Sir David Lane, Cancer Research UK | Tamoxifen has been a huge success story helping to prevent breast cancer recurring for many women Professor Sir David Lane, Cancer Research UK |
Which molecule wins determines if that switch is off or on. | Which molecule wins determines if that switch is off or on. |
Dr Jason Carroll, who led the study, said: "We knew that women developed resistance to tamoxifen but previously our understanding of why this occurred could be compared with trying to fix a broken car without knowing how the engine worked. | Dr Jason Carroll, who led the study, said: "We knew that women developed resistance to tamoxifen but previously our understanding of why this occurred could be compared with trying to fix a broken car without knowing how the engine worked. |
"Now we understand how all the engine parts operate and we can try to think about ways to make repairs." | "Now we understand how all the engine parts operate and we can try to think about ways to make repairs." |
He added: "We can use this information to predict who will respond to tamoxifen and, more importantly, who won't. | He added: "We can use this information to predict who will respond to tamoxifen and, more importantly, who won't. |
"It will mean that we would no longer waste time that could have been better used giving more effective therapies and treatments. | "It will mean that we would no longer waste time that could have been better used giving more effective therapies and treatments. |
Test hope | Test hope |
If a woman is not going to benefit from tamoxifen, she could be given other drugs such as Herceptin or a class of medicines called aromatase inhibitors, which act on tumours in different ways. | If a woman is not going to benefit from tamoxifen, she could be given other drugs such as Herceptin or a class of medicines called aromatase inhibitors, which act on tumours in different ways. |
Dr Carroll said the failed mechanism would not account for all cases of tamoxifen resistance. | Dr Carroll said the failed mechanism would not account for all cases of tamoxifen resistance. |
But he added: "We're not talking about a small percentage of cases of tamoxifen resistance. I would think it's going to account for quite a significant number." | But he added: "We're not talking about a small percentage of cases of tamoxifen resistance. I would think it's going to account for quite a significant number." |
The researchers say it is important for their findings to be replicated in larger groups. | |
But they say a test could be possible in five years' time, and that the process that stops tamoxifen working could also occur with other drugs. | |
Professor Sir David Lane, Cancer Research UK's chief scientist said: "Tamoxifen has been a huge success story helping to prevent breast cancer recurring for many women. | Professor Sir David Lane, Cancer Research UK's chief scientist said: "Tamoxifen has been a huge success story helping to prevent breast cancer recurring for many women. |
"Understanding why it occasionally stops working is really important because it allows us to identify new targets for drug development and who will need such treatments." | "Understanding why it occasionally stops working is really important because it allows us to identify new targets for drug development and who will need such treatments." |
Dr Alexis Willett, of Breakthrough Breast Cancer, said: "This research gives us a better understanding of one of the ways resistance can occur and is an important step towards developing improved treatments for patients. | Dr Alexis Willett, of Breakthrough Breast Cancer, said: "This research gives us a better understanding of one of the ways resistance can occur and is an important step towards developing improved treatments for patients. |
"It's vital that research continues into why resistance occurs and how to overcome it." | "It's vital that research continues into why resistance occurs and how to overcome it." |
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